16
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T62611 | Adenosine receptor antagonist 2 | ||
Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects. | |||
T21620 | Adenosine receptor antagonist 4 | Adenosine Receptor | |
Adenosine receptor antagonist 4 is an adenosine receptor antagonist. | |||
T37793 | A2B receptor antagonist 2 | A2B receptor antagonist 2 | Adenosine Receptor |
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B). | |||
T77508 | A2B receptor antagonist 2 hydrochloride | ||
A2B receptor antagonist 2 hydrochloride is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B). | |||
T22031 | ANR 94 | Adenosine Receptor | |
ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows promise for research into Parkinson's disease. [1] [2] | |||
T16811 | RWJ-51204 | GABA Receptor | |
RWJ-51204 is a selective adenosine A2A receptor antagonist and a partial agonist of GABA(A) receptor (IC50: 0.2-2 nM). It has neuroprotective and movement-improving effects and can be used in research related to Parkinso... | |||
T25840 | MSX-2 | MSX 2 | |
MSX-2 is an A2A adenosine receptor antagonist. | |||
T25841 | MSX-3 | MSX 3 | |
MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2. | |||
T63326 | A2A receptor antagonist 2 | ||
A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM). | |||
T69566 | MSX-3 free acid | ||
MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2. | |||
T72588 | A3AR antagonist 2 | ||
A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM. | |||
T60580 | A1AR antagonist 2 | ||
A1AR antagonist 2 (compound 18h) is a potent antagonist of the A1 adenosine receptor (AR). A1AR antagonist 2 has Ki values of 1.49, 10.2, and 50.1 nM for hA 1, hA 2A, and hA 2B, respectively [1]. | |||
T70770 | Cyclazosin Free Base | ||
Cyclazosin Free Base is a monocarboxylic acid amide obtained by formal condensation of the carboxy group of furoic acid with the secondary amino group of 6,7-dimethoxy-2-[(4aR,8aS)-octahydroquinoxalin-1-yl]quinazolin-4-a... | |||
T72626 | A2AR-antagonist-1 | Adenosine Receptor | |
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability in mouse liver microsomes (t1/2 = 86.1 min). Additionally,... | |||
T60511 | Theophylline sodium glycinate | ||
Theophylline (1,3-Dimethylxanthine) sodium glycinate is a potent inhibitor of phosphodiesterase (PDE) that inhibits PDE3 activity to relax airway smooth muscle. Theophylline sodium glycinate can be used for the research ... | |||
T36679 | Rp-cAMPS sodium salt | ||
Rp-cAMPS sodium salt, a cAMP analog, is a potent, competitive cAMP-induced activation of cAMP-dependent PKA I and II (Kis of 12.5 μM and 4.5 μM, respectively) antagonist. Rp-cAMPS sodium salt is resistant to hydrolysis b... |