Home Tools
Log in
Cart

Search Result

Search Results for " adenosine receptor antagonist 2 "

16

Compounds

Cat No. Product Name Synonyms Targets
T62611 Adenosine receptor antagonist 2
Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
T21620 Adenosine receptor antagonist 4 Adenosine Receptor
Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
T37793 A2B receptor antagonist 2 A2B receptor antagonist 2 Adenosine Receptor
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T77508 A2B receptor antagonist 2 hydrochloride
A2B receptor antagonist 2 hydrochloride is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T22031 ANR 94 Adenosine Receptor
ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows promise for research into Parkinson's disease. [1] [2]
T16811 RWJ-51204 GABA Receptor
RWJ-51204 is a selective adenosine A2A receptor antagonist and a partial agonist of GABA(A) receptor (IC50: 0.2-2 nM). It has neuroprotective and movement-improving effects and can be used in research related to Parkinso...
T25840 MSX-2 MSX 2
MSX-2 is an A2A adenosine receptor antagonist.
T25841 MSX-3 MSX 3
MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.
T63326 A2A receptor antagonist 2
A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).
T69566 MSX-3 free acid
MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.
T72588 A3AR antagonist 2
A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.
T60580 A1AR antagonist 2
A1AR antagonist 2 (compound 18h) is a potent antagonist of the A1 adenosine receptor (AR). A1AR antagonist 2 has Ki values of 1.49, 10.2, and 50.1 nM for hA 1, hA 2A, and hA 2B, respectively [1].
T70770 Cyclazosin Free Base
Cyclazosin Free Base is a monocarboxylic acid amide obtained by formal condensation of the carboxy group of furoic acid with the secondary amino group of 6,7-dimethoxy-2-[(4aR,8aS)-octahydroquinoxalin-1-yl]quinazolin-4-a...
T72626 A2AR-antagonist-1 Adenosine Receptor
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability in mouse liver microsomes (t1/2 = 86.1 min). Additionally,...
T60511 Theophylline sodium glycinate
Theophylline (1,3-Dimethylxanthine) sodium glycinate is a potent inhibitor of phosphodiesterase (PDE) that inhibits PDE3 activity to relax airway smooth muscle. Theophylline sodium glycinate can be used for the research ...
T36679 Rp-cAMPS sodium salt
Rp-cAMPS sodium salt, a cAMP analog, is a potent, competitive cAMP-induced activation of cAMP-dependent PKA I and II (Kis of 12.5 μM and 4.5 μM, respectively) antagonist. Rp-cAMPS sodium salt is resistant to hydrolysis b...
TargetMol